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TGR-1202 hydrochloride
TGR-1202 hydrochloride
会员等级价V
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  • 商品货号:A16278
  • 名称:TGR-1202 hydrochloride
  • 简介:TGR-1202 hydrochloride is an orally available, next generation PI3Kδ inhibitor, inhibits PI3Kδ activity in enzyme and cell based assays with IC50 and EC50 values of 22.2 and 24.3 nM respectively.
  • CASNO:1532533-78-0
  • 分子式:C31H25ClF3N5O3
  • 分子量:608.01
  • SMILES:O=C1C(C2=CC=CC(F)=C2)=C([C@@H](N3N=C(C4=CC=C(OC(C)C)C(F)=C4)C5=C(N)N=CN=C53)C)OC6=CC=C(F)C=C16.[H]Cl
  • 保持条件:at -20°C 3 years Powder
  • 同名:RP5264 hydrochloride, TGR1202 hydrochloride, TGR 1202 hydrochloride, RP-5264 hydrochloride, RP 5264 hydrochloride
  • 纯度:>98%
  • 应用:PI3Kδ inhibitor
  • 作用机制:Inhibitor