• 名称：RQ-00203078
• 简介：RQ-00203078 is a highly selective, potent and orally available TRPM8 antagonist (IC50 values are 5.3 and 8.3 nM for rat and human channels respectively), exhibits >350-fold selectivity for TRPM8 over TRPV4, TRPV1 and TRPA1.
• CASNO：1254205-52-1
• 分子式：C21H13ClF6N2O5S
• 分子量：554.85
• SMILES：ClC1=C(N(CC2=CC=C(OC(F)(F)F)C=C2)S(C3=CC=C(C(O)=O)C=C3)(=O)=O)N=CC(C(F)(F)F)=C1
• 保持条件：at -20°C 3 years Powder
• 同名：RQ 00203078, RQ00203078
• 纯度：>98%
• 应用：TRPM8 antagonist
• 作用机制：Antagonist