- 名称:TAPI-2
- 简介:TAPI-2 is an inhibitor of TACE, ADAMs, ACE secretase, and other MMPs (metalloproteinases). TAPI-2 blocks release of DCC7, APP, TNFα, L-selectin, NOTCH, TGFα, IL-6R9, erbB2/HER2, and ACE. This inhibitor has been used in tissue culture.
- CASNO:187034-31-7
- 分子式:C19H37N5O5
- 分子量:415.53
- SMILES:C[C@@H](C(=O)NCCN)NC(=O)[C@H](C(C)(C)C)NC(=O)C(CC(C)C)CC(=O)NO
- 保持条件:at -20°C 3 years Powder
- 同名:TNF Protease Inhibitor 2
- 纯度:>98%
- 应用:TACE/MMP inhibitor
- 作用机制:Inhibitor