- 名称:NPS-2143 (SB-262470)
- 简介:NPS-2143 is a selective Ca2+-sensing receptor antagonist, shown to block increases in cytoplasmic Ca2+ concentrations elicited by human Ca2+ receptors expressed in HEK293 cells with an IC50 of 43 nM.
- CASNO:284035-33-2
- 分子式:C24H25ClN2O2
- 分子量:408.9
- SMILES:CC(C)(CC1=CC2=CC=CC=C2C=C1)NC[C@H](COC3=C(C(=CC=C3)Cl)C#N)O
- 保持条件:at -20°C 3 years Powder
- 同名:NPS2143, SB262470
- 纯度:>98%
- 应用:CaSR antagonist
- 作用机制:Antagonist