- 商品货号:A14133
- 名称:GSK1324726A (I-BET726)
- 简介:GSK1324726A (I-BET726) is a novel, potent, and selective small molecule inhibitor of BET proteins with high affinity to BRD2 (IC50= 41 nM), BRD3 (IC50= 31 nM), and BRD4 (IC50= 22 nM).
- CASNO:1300031-52-0
- 分子式:C25H23ClN2O3
- 分子量:434.91
- SMILES:CC1CC(C2=C(N1C(=O)C)C=CC(=C2)C3=CC=C(C=C3)C(=O)O)NC4=CC=C(C=C4)Cl
- 保持条件:at -20°C 3 years Powder
- 同名:I-BET726, GSK 1324726A, GSK-1324726A, I-BET 726
- 纯度:>98%
- 应用:BET inhibitor
- 作用机制:Inhibitor